1. 2024
  2. A synthesis of novel 5-methylsulfanylazolo[1,5-a]pyrimidin-7(4H)-ones and investigation of their chemical and cytotoxic properties

    Lyapustin, D., Fayzullina, D., Marusich, I., Kotovskaya, S., Melekhin, V., Tokhtueva, M., Ulomsky, E. & Rusinov, V., 1 Feb 2024, In: Chemistry of Heterocyclic Compounds. 60, 1-2, p. 52-57 6 p.

    Research output: Contribution to journalArticlepeer-review

  3. 2023
  4. 5-Alkylamino-7-aminoazolo[1,5-a]pyrimidine-6-carbonitriles: synthetic strategies and anticancer activity in vitro

    Urakov, G. V., Savateev, K. V., Melekhin, V. V., Kotovskaya, S. K. & Rusinov, V. L., 1 Dec 2023, In: Russian Chemical Bulletin. 72, 12, p. 3022-3031 10 p.

    Research output: Contribution to journalArticlepeer-review

  5. Диметил 7-метил-2-n-толил-4-фенилпирроло[2,1-f] [2,1,4]триазин-5,6-дикарбоксилат, обладающий антикоагулянтным действием: патент на изобретение

    Мочульская, Н. Н., Котовская, С. К., Русинов, В. Л., Чарушин, В. Н., Спасов, А. А., Кучерявенко, А. Ф. & Гайдукова, К. А., 17 Feb 2023, IPC No. C07D 487/04, C07D 519/00, A61K 31/53, A61P 7/02, Федеральный институт промышленной собственности, Patent No. 2790375, 22 Mar 2022, Priority date 22 Mar 2022, Priority No. 2022107619

    Research output: Patent

  6. Bioactive Pyrrolo[2,1-f][1,2,4]triazines: Synthesis, Molecular Docking, In Vitro Cytotoxicity Assay and Antiviral Studies

    Mochulskaya, N. N., Kotovskaya, S. K., Butorin, I. I., Varaksin, M. V., Charushin, V. N., Rusinov, V. L., Esaulkova, Y. L., Slita, A. V., Ilyina, P. A. & Zarubaev, V. V., 2023, In: Chemistry (Switzerland). 5, 4, p. 2657-2676 20 p.

    Research output: Contribution to journalArticlepeer-review

  7. Synthesis and cytotoxic activity of (2-arylquinazolin-4-yl)hydrazones of 2-hydroxybenzaldehydes

    Nosova, E. V., Butorin, I. I., Likhacheva, M. D. & Kotovskaya, S. K., 2023, In: Chimica Techno Acta. 10, 2, 202310211.

    Research output: Contribution to journalArticlepeer-review

  8. 2022
  9. 6-(Tetrazol-5-yl)-7-aminoazolo[1,5-a]pyrimidines as Novel Potent CK2 Inhibitors

    Urakov, G. V., Savateev, K. V., Kotovskaya, S. K., Rusinov, V. L., Spasov, A. A., Babkov, D. A. & Sokolova, E. V., 7 Dec 2022, In: Molecules. 27, 24, 8697.

    Research output: Contribution to journalArticlepeer-review

  10. The Effects of Nitroazolopyrimidines on the A1 Adenosine Receptor and Intraocular Pressure in Rats

    Savateev, K. V., Rusinov, V. L., Kotovskaya, S. K., Spasov, A. A., Naumenko, L. V., Taran, A. S., Brigadirova, A. A., Yakovlev, D. S., Sultanova, K. T. & Shcherbakova, N. M., 1 Aug 2022, In: Russian Journal of Bioorganic Chemistry. 48, 4, p. 777-782 6 p.

    Research output: Contribution to journalArticlepeer-review

  11. CK2 Inhibition and Antitumor Activity of 4,7-Dihydro-6-nitroazolo[1,5-a]pyrimidines

    Lyapustin, D. N., Kotovskaya, S. K., Butorin, I. I., Ulomsky, E. N., Rusinov, V. L., Babkov, D. A., Pokhlebin, A. A., Spasov, A. A., Melekhin, V. V., Tokhtueva, M. D., Shcheglova, A. V. & Makeev, O. G., Aug 2022, In: Molecules. 27, 16, 5239.

    Research output: Contribution to journalArticlepeer-review

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